Diltiazem is a Calcium Channel Blocker (CCB) and it can interact significantly with drugs such as Cisapride, Colchicine, Lomitapide, Eryhthromycin, Amiodarone, Clopidogrel, Beta Blockers, Droperidol, Dantrolene, Lacosamide, Clonidine, Fingolimod, CYP3A4 inhibitors (Clarithromycin, Ceritinib, Atazanavir, etc.), CYP3A4 inducers (Carbamazepine, St.John’s wort, etc.), CYP3A4 substrates (Simvastatin, Atorvastatin, Lovastatin, Apixaban, Domperidone, Donepezil, Dronedarone, Clozapine, Fentanyl, Hydrocodone, Piperaquine, Erlotinib, Nilotinib, Crizotinib, Bosutinib, Ibratinib, Doxorubicin, Simeprevir, Lurasidone, Ranolazine, Eplerenone, Everolimus, Aripiprazole, Eliglustat, Cilostazol, Tolvaptan, Ivabradine, etc.) and P-gp substrates (Dabigatran, Apixaban, Everolimus, Vincristine, Nilotinib, Afatinib, Bosutinib, Trabectedin, Ombitasvir, Simeprevir, Dasabuvir, Paritaprevir, Topotecan, etc.).
Tags:
Calcium channel blocker , CYP3A4 inducers , CYP3A4 inhibitors , Drug Interactions of Diltiazem , P-gp substrates
By:
nainamohamedpakk
Education
65 months ago
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