Narrated ADHD

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Ch. 36

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Chapter 36: 

Chapter 36 Central Nervous System Stimulants and Attention-Deficit/Hyperactivity Disorder

CNS Stimulants: 

CNS Stimulants Increase the activity of CNS neurons Enhance the neuronal excitation; a few suppress the neuronal inhibition In sufficient doses, all can cause convulsions Limited clinical applications

CNS Stimulants and Attention-Deficit/Hyperactivity Disorder: 

CNS Stimulants and Attention-Deficit/Hyperactivity Disorder Amphetamines Methyphenidate and dexmethylphenidate Methylxanthines Miscellaneous stimulants Attention-deficit/hyperactivity disorder (ADHD)

Amphetamines: 

Amphetamines Pharmacologic effects Central nervous system Cardiovascular system Tolerance With regular use, develops to elevation of mood, suppression of appetite, and stimulation of the heart and blood vessels Physical dependence Abstinence syndrome with abrupt withdrawal Abuse High potential for abuse due to euphoria

Amphetamines: 

Amphetamines Adverse effects CNS stimulation Weight loss Cardiovascular effects Psychosis

Amphetamines: 

Amphetamines Toxicity Dysrhythmias Hypertension Dizziness Confusion Hallucinations Convulsions Paranoid delusions Coma Palpitations Cerebral hemorrhage

Amphetamines: 

Amphetamines Treatment Chlorpromazine Alpha-adrenergic blocker Diazepam Therapeutic uses ADHD Narcolepsy Obesity (not recommended due to risk for abuse)

Amphetamines: 

Amphetamines Preparations, dosage, and administration Dextroamphetamine sulfate Short duration (Dexedrine, Dextrostat) Long duration (Dexedrine Spansules) Amphetamine/dextroamphetamine mixture Short duration (Adderall) Long duration (Adderall-XR) Methamphetamine (Desoxyn)

Methylphenidate: 

Methylphenidate Trade names Ritalin, Metadate, Methylin, Concerta 50:50 mixture of dextro and levo isomers Preparations, dosage, and administration Short duration Ritalin, Methylin Intermediate duration Ritalin SR, Metadate ER, Methylin ER Long duration Concerta, Metadate CD, Ritalin LA

Methylxanthines: 

Methylxanthines Derivates of xanthine Caffeine Few clinical applications Widespread ingestion for nonmedical purposes Dietary sources Chocolate Desserts Soft drinks Cola nut

Methylxanthines: 

Methylxanthines Mechanism of action Reversible blockade of adenosine receptors Calcium permeability Accumulation of cyclic AMP Low doses Decreases drowsiness and fatigue and increases capacity for prolonged intellectual exertion Increasing doses Nervousness, insomnia, tremors Seizures with very large amounts

Methylxanthines: 

Methylxanthines Pharmacologic effects Central nervous system Heart Blood vessels Bronchi Kidney Reproduction Pharmacokinetics Readily absorbed from the GI tract Achieves peak plasma levels within 1 hour Eliminated by hepatic metabolism

Methylxanthines: 

Methylxanthines Therapeutic uses Neonatal apnea Promoting wakefulness Other applications Acute toxicity Stimulation of the CNS Tachycardia Respiratory stimulation Sensory phenomena

Methylxanthines: 

Methylxanthines Preparations, dosage, and administration For promoting wakefulness For neonatal apnea Theophylline Theobromine

Attention-Deficit/Hyperactivity Disorder (ADHD) in Children: 

Attention-Deficit/Hyperactivity Disorder (ADHD) in Children Signs and symptoms Inattention Hyperactivity Impulsivity Fidgety Unable to concentrate

ADHD in Children: 

ADHD in Children Signs and symptoms (cont ’ d) Unable to wait his or her turn Switches excessively from one activity to another Calls out excessively in class Present prior to age 7 years Present for at least 6 months

ADHD in Children: 

ADHD in Children Etiology Management overview Cognitive therapy Stimulant drugs Drug therapy I: CNS stimulants Methylphenidate (Ritalin, Concerta, others) Dexmethylphenidate (Focalin) Dextroamphetamine (Dexedrine, others) Amphetamine mixture (Adderall) Pemoline (Cylert)

ADHD in Children: 

ADHD in Children Drug therapy II: atomoxetine Description and therapeutic effects Nonstimulant No potential for abuse Administered once a day

ADHD in Children: 

ADHD in Children Drug therapy II: atomoxetine Adverse effects GI reactions Reduced appetite Dizziness Somnolence Mood swings Trouble sleeping

ADHD in Children: 

ADHD in Children Drug therapy II: atomoxetine (cont ’ d) Drug interactions MAO inhibitors (isocarboxazid, phenelzine) CYP2D6 (paroxetine, fluoxetine, quinidine) Role in ADHD therapy Preparations, dosage, and administration Children who weigh less than 70 kg Children who weigh more than 70 kg

ADHD in Children: 

ADHD in Children Drug therapy III: antidepressants Tricycle antidepressants Decrease hyperactivity Little effect on impulsivity and inattention Second-line drugs Bupropion (Wellbutrin) Can reduce behavioral symptoms Less effective than stimulants Poses risk of seizure Second-line drug

ADHD in Adults: 

ADHD in Adults Drug therapy III: antidepressants 60% of ADHD cases persist into adulthood Symptoms Poor concentration Stress intolerance Antisocial behavior Outbursts of anger Inability to maintain a routine Drug therapy Methylphenidate