logging in or signing up Pharmacology aSGuest1040 Download Post to : URL : Related Presentations : Share Add to Flag Embed Email Send to Blogs and Networks Add to Channel Uploaded from authorPOINT lite Insert YouTube videos in PowerPont slides with aS Desktop Copy embed code: (To copy code, click on the text box) Embed: URL: Thumbnail: WordPress Embed Customize Embed The presentation is successfully added In Your Favorites. Views: 2585 Category: Science & Tech.. License: All Rights Reserved Like it (0) Dislike it (0) Added: October 15, 2008 This Presentation is Public Favorites: 2 Presentation Description No description available. Comments Posting comment... By: kokooo (32 month(s) ago) it is a great pp Saving..... Post Reply Close Saving..... Edit Comment Close Premium member Presentation Transcript Pharmacology : Pharmacology Drugs that Affect the Endocrine System Topics : Topics Pituitary Drugs Parathyroid/Thyroid Drugs Adrenal Drugs Pancreatic Drugs Reproductive Drugs Sexual Behavior Drugs Functions : Functions Regulation Control Glands : Glands Exocrine Secrete enzymes Close to organs Endocrine Secrete hormones Transport via bloodstream Require receptors Slide 5: Nervous Endocrine Mechanism of Action : Mechanism of Action Hypothalamus : Hypothalamus Hypothalamic Control Pituitary : Hypothalamic Control Pituitary Posterior Pituitary : Posterior Pituitary Anterior Pituitary : Anterior Pituitary Anterior Pituitary : Anterior Pituitary Anterior Pituitary : Anterior Pituitary Pituitary Hormones : Pituitary Hormones Thyroid : Thyroid Thyroid : Thyroid Hypothyroidism : Hypothyroidism Hyperthyroidism : Hyperthyroidism Parathyroid : Parathyroid Parathyroid : Parathyroid Calcium Regulation : Calcium Regulation Pancreas : Pancreas Pancreas : Pancreas Alpha cells: glucagon Beta cells: insulin Pancreas : Pancreas Glucose Regulation : Glucose Regulation Adrenal : Adrenal Adrenal Medulla : Adrenal Medulla Adrenal Cortex : Adrenal Cortex Anterior Pituitary Drugs : Anterior Pituitary Drugs Inadequate Growth Hormone Dwarfism somatrem (Protropin®) homatropin (Humatrope®) Excessive Growth Hormone Acromegaly Gigantism Surgical removal 1º octreotide (Sandostatin®) Posterior Pituitary Drugs : Posterior Pituitary Drugs Oxytocin ADH Diabetes insipidus Nocturnal enuresis vasopressin (Pitressin®) desmopressin (Stimate®) lypressin (Diapid®) Parathyroid Diseases : Parathyroid Diseases Hypoparathyroidism Inadequate calcium levels TX: increased dietary calcium Hyperparathyroidism Excessive calcium levels TX: surgical removal Thyroid Disease : Thyroid Disease Hypothyroidism Hormone replacement levothyroxine (Synthroid®) Hyperthyroidism Thyrotoxicosis Surgical removal propylthiouracil (PTU) Adrenal Cortex : Adrenal Cortex ACTH Hypersecretion Cushing’s Disease Surgical removal Inhibit adrenal secretion ketoconazol (Nizoral ®) Symptomatic tx: Antihypertensives ACTH Hyposecretion Addison’s Disease Replacement therapy Cortisone (Cortistan®) Hydrocortisone (SoluCortef®) Fludrocortisone (Florinef Acetate®) Pancreas : Pancreas Insulin Preparations : Insulin Preparations Regular Insulin Natural insulin Modified Insulin Increased duration of action NPH (neutral protamin Hagedorn) Natural plus protamin Lente Attached to zinc to prolong absorption Oral Hypoglycemic Agents : Oral Hypoglycemic Agents Sulfonylureas insulin secretion tolbutamide (Orinase®) chlorpropamide (Diabinese®) glipizide (Glucotrol®) glyburide (Micronase®) Alpha-glucosidase inhibitors Delay carbohydrate metabolism acarbose (Precose®) miglitol (Glyset®) Biguanides metformin (Glucophage®) Glucose synthesis Glucose uptake Thiazolidinediones Insulin effectiveness troglitazone (Rezulin®) Hyperglycemic Agents : Hyperglycemic Agents Glucagon gluconeogenesis D50W diazoxide (Proglycem®) Inhibits insulin release Estrogens & Progestins : Estrogens & Progestins Estrogens used for post-menopausal hormone replacement therapy. estradiol (Estrace®) conjugated estrogens (Premarin®) estropipate (Ogen®) Progestin Diminish side effects of estrogen therapy Nausea, fluid retention, breast tenderness medroxyprogesterone acetate (Provera®) norethindrone acetate (Aygestin®) Oral Contraceptives : Oral Contraceptives Combination of estrogen and progestin Loestrin®, Levora®, Nordette®, Ovocon®, Norinyl® plus many others Minipill: progestin only Micronor®, Nor-Q.D.®, Orvette® Prime side effect: risk of thromboembolism Uterine Stimulants & Relaxants : Uterine Stimulants & Relaxants Stimulants (Oxytocics) uterine contraction Indication: Induce labor Postpartum hemorrhage oxytocin (Pitocin®) ergonovine (Ergotrate®) Relaxants (tocolytics) Relax uterine smooth muscle Beta2 agonists terbutaline (Brethine®) ritodrine (Yuptopar®) Infertility Agents : Infertility Agents Promote maturation of ovarian follicles clomiphene (Clomid®) urofollitropin (Metrodin®) Male Reproductive Agents : Male Reproductive Agents Testosterone Replacement methyltestosterone (Metandren®) fluoxymesterone (Halotestin®) Benign Prostatic Hypertrophy Surgery finasteride (Proscar®) Sexual Behavior : Sexual Behavior Most are side effects from other medications Antihypertensives & psychoactive drugs sildenafil (Viagra®) You do not have the permission to view this presentation. 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Pharmacology aSGuest1040 Download Post to : URL : Related Presentations : Share Add to Flag Embed Email Send to Blogs and Networks Add to Channel Uploaded from authorPOINT lite Insert YouTube videos in PowerPont slides with aS Desktop Copy embed code: (To copy code, click on the text box) Embed: URL: Thumbnail: WordPress Embed Customize Embed The presentation is successfully added In Your Favorites. Views: 2585 Category: Science & Tech.. License: All Rights Reserved Like it (0) Dislike it (0) Added: October 15, 2008 This Presentation is Public Favorites: 2 Presentation Description No description available. Comments Posting comment... By: kokooo (32 month(s) ago) it is a great pp Saving..... Post Reply Close Saving..... Edit Comment Close Premium member Presentation Transcript Pharmacology : Pharmacology Drugs that Affect the Endocrine System Topics : Topics Pituitary Drugs Parathyroid/Thyroid Drugs Adrenal Drugs Pancreatic Drugs Reproductive Drugs Sexual Behavior Drugs Functions : Functions Regulation Control Glands : Glands Exocrine Secrete enzymes Close to organs Endocrine Secrete hormones Transport via bloodstream Require receptors Slide 5: Nervous Endocrine Mechanism of Action : Mechanism of Action Hypothalamus : Hypothalamus Hypothalamic Control Pituitary : Hypothalamic Control Pituitary Posterior Pituitary : Posterior Pituitary Anterior Pituitary : Anterior Pituitary Anterior Pituitary : Anterior Pituitary Anterior Pituitary : Anterior Pituitary Pituitary Hormones : Pituitary Hormones Thyroid : Thyroid Thyroid : Thyroid Hypothyroidism : Hypothyroidism Hyperthyroidism : Hyperthyroidism Parathyroid : Parathyroid Parathyroid : Parathyroid Calcium Regulation : Calcium Regulation Pancreas : Pancreas Pancreas : Pancreas Alpha cells: glucagon Beta cells: insulin Pancreas : Pancreas Glucose Regulation : Glucose Regulation Adrenal : Adrenal Adrenal Medulla : Adrenal Medulla Adrenal Cortex : Adrenal Cortex Anterior Pituitary Drugs : Anterior Pituitary Drugs Inadequate Growth Hormone Dwarfism somatrem (Protropin®) homatropin (Humatrope®) Excessive Growth Hormone Acromegaly Gigantism Surgical removal 1º octreotide (Sandostatin®) Posterior Pituitary Drugs : Posterior Pituitary Drugs Oxytocin ADH Diabetes insipidus Nocturnal enuresis vasopressin (Pitressin®) desmopressin (Stimate®) lypressin (Diapid®) Parathyroid Diseases : Parathyroid Diseases Hypoparathyroidism Inadequate calcium levels TX: increased dietary calcium Hyperparathyroidism Excessive calcium levels TX: surgical removal Thyroid Disease : Thyroid Disease Hypothyroidism Hormone replacement levothyroxine (Synthroid®) Hyperthyroidism Thyrotoxicosis Surgical removal propylthiouracil (PTU) Adrenal Cortex : Adrenal Cortex ACTH Hypersecretion Cushing’s Disease Surgical removal Inhibit adrenal secretion ketoconazol (Nizoral ®) Symptomatic tx: Antihypertensives ACTH Hyposecretion Addison’s Disease Replacement therapy Cortisone (Cortistan®) Hydrocortisone (SoluCortef®) Fludrocortisone (Florinef Acetate®) Pancreas : Pancreas Insulin Preparations : Insulin Preparations Regular Insulin Natural insulin Modified Insulin Increased duration of action NPH (neutral protamin Hagedorn) Natural plus protamin Lente Attached to zinc to prolong absorption Oral Hypoglycemic Agents : Oral Hypoglycemic Agents Sulfonylureas insulin secretion tolbutamide (Orinase®) chlorpropamide (Diabinese®) glipizide (Glucotrol®) glyburide (Micronase®) Alpha-glucosidase inhibitors Delay carbohydrate metabolism acarbose (Precose®) miglitol (Glyset®) Biguanides metformin (Glucophage®) Glucose synthesis Glucose uptake Thiazolidinediones Insulin effectiveness troglitazone (Rezulin®) Hyperglycemic Agents : Hyperglycemic Agents Glucagon gluconeogenesis D50W diazoxide (Proglycem®) Inhibits insulin release Estrogens & Progestins : Estrogens & Progestins Estrogens used for post-menopausal hormone replacement therapy. estradiol (Estrace®) conjugated estrogens (Premarin®) estropipate (Ogen®) Progestin Diminish side effects of estrogen therapy Nausea, fluid retention, breast tenderness medroxyprogesterone acetate (Provera®) norethindrone acetate (Aygestin®) Oral Contraceptives : Oral Contraceptives Combination of estrogen and progestin Loestrin®, Levora®, Nordette®, Ovocon®, Norinyl® plus many others Minipill: progestin only Micronor®, Nor-Q.D.®, Orvette® Prime side effect: risk of thromboembolism Uterine Stimulants & Relaxants : Uterine Stimulants & Relaxants Stimulants (Oxytocics) uterine contraction Indication: Induce labor Postpartum hemorrhage oxytocin (Pitocin®) ergonovine (Ergotrate®) Relaxants (tocolytics) Relax uterine smooth muscle Beta2 agonists terbutaline (Brethine®) ritodrine (Yuptopar®) Infertility Agents : Infertility Agents Promote maturation of ovarian follicles clomiphene (Clomid®) urofollitropin (Metrodin®) Male Reproductive Agents : Male Reproductive Agents Testosterone Replacement methyltestosterone (Metandren®) fluoxymesterone (Halotestin®) Benign Prostatic Hypertrophy Surgery finasteride (Proscar®) Sexual Behavior : Sexual Behavior Most are side effects from other medications Antihypertensives & psychoactive drugs sildenafil (Viagra®)